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Clinical Trial Details — Status: Completed

Administrative data

NCT number NCT01862081
Other study ID # GO27802
Secondary ID 2013-003543-28
Status Completed
Phase Phase 1
First received May 22, 2013
Last updated November 27, 2017
Start date July 16, 2013
Est. completion date June 9, 2017

Study information

Verified date November 2017
Source Genentech, Inc.
Contact n/a
Is FDA regulated No
Health authority
Study type Interventional

Clinical Trial Summary

This is an open-label, multicenter, dose-escalation study designed to assess the safety, tolerability, and pharmacokinetics of oral GDC-0032 administered in combination with either docetaxel or with paclitaxel. Patients treated with the GDC-0032 and docetaxel have HER2-negative locally recurrent or metastatic breast cancer or non-small cell lung cancer (NSCLC). Patients treated with the GDC-0032 and paclitaxel combination have human epidermal growth factor receptor 2 (HER2)-negative locally recurrent or metastatic breast cancer. There are two potential stages within each arm of this study: a dose-escalation stage (Stage 1) and a dose-expansion stage (Stage 2). Once the maximum tolerated dose of GDC-0032 in a given arm has been established from dose escalation, additional patients with each combination will be enrolled in Stage 2.


Recruitment information / eligibility

Status Completed
Enrollment 80
Est. completion date June 9, 2017
Est. primary completion date June 9, 2017
Accepts healthy volunteers No
Gender All
Age group 18 Years and older
Eligibility Inclusion Criteria:

- Age >=18 years

- For paclitaxel combination arms: histologically or cytologically documented adenocarcinoma of the breast with locally recurrent or metastatic disease

- For docetaxel combination arms: histologically or cytologically documented adenocarcinoma of the breast with locally recurrent or metastatic disease or histologically documented advanced (Stage IV) or recurrent NSCLC

- For participants with breast cancer: HER2-negative disease as defined by local clinical guidelines

- Participants with NSCLC to be treated with docetaxel need to have received at least one prior anti-cancer treatment regimen in an advanced setting and to have docetaxel be considered appropriate treatment

- Evaluable or measurable disease per response evaluation criteria in solid tumors (RECIST) v.1.1

- Life expectancy >=12 weeks

- Eastern cooperative oncology group (ECOG) performance status of 0 or 1 at screening

- Adequate hematologic and end organ function

- Use of highly effective form of contraception

Exclusion Criteria:

- Prior anti-cancer therapy

- Prior treatment with phosphoinositide 3-kinase (PI3K) inhibitor

- Known significant hypersensitivity to any components of study treatment

- Grade >=2 peripheral neuropathy

- Type 1 or Type 2 diabetes

- Grade >=2 hypercholesterolemia or hypertriglyceridemia

- Congenital long QT syndrome

- Active congestive heart failure or ventricular arrhythmia

Study Design


Intervention

Drug:
Docetaxel
Participants will receive docetaxel 75 milligrams per meter-squared (mg/m^2) intravenous (IV) dose on Day 1 of each 21-day cycle.
GDC-0032
Participants will receive escalated dose of GDC-0032. The initial dose will be 3 mg capsules or 2 mg tablets.
Paclitaxel
Participants will receive paclitaxel 80 mg/m^2 IV dose on Day 1, 8, 15 and 22 of each 28-day cycle.

Locations

Country Name City State
Belgium UZ Leuven; Maag, -darm en leverziekten/endoscopie - Endoscopy Leuven
Canada Princess Margaret Hospital Toronto Ontario
Spain Hospital Universitari Vall d'Hebron Barcelona
Spain Hospital Clinico Universitario de Valencia Valencia
United States Dana Farber Cancer Institute Boston Massachusetts
United States Massachusetts General Hospital Boston Massachusetts
United States Texas Oncology, P.A; Baylor Sammons Cancer Center Dallas Texas
United States Barbara Ann Karmanos Cancer Institute Detroit Michigan
United States Texas Oncology, P.A. - Fort Worth Fort Worth Texas
United States Sarah Cannon Research Institute Nashville Tennessee
United States Vanderbilt University Medical Center Nashville Tennessee
United States Virginia Oncology Associates Norfolk Virginia
United States Florida Cancer Specialists - Tampa (Dr. MLK Blvd) Tampa Florida
United States Yakima Valley Memorial Hospital/North Star Lodge Yakima Washington

Sponsors (1)

Lead Sponsor Collaborator
Genentech, Inc.

Countries where clinical trial is conducted

United States,  Belgium,  Canada,  Spain, 

Outcome

Type Measure Description Time frame Safety issue
Primary Safety: Incidence of adverse events Approximately 3 years
Primary Safety: Incidence of dose limiting toxicities Up to 28 days
Secondary Area under the curve from time 0 to the last measurable concentration (AUC0-last) Up to 28 days
Secondary Time to maximum observed plasma concentration (Tmax) Up to 28 days
Secondary Maximum observed plasma concentration (Cmax) Up to 28 days
Secondary Minimum observed plasma concentration (Cmin) Up to 28 days
Secondary Objective response according to RECIST v1.1 Approximately 3 years
Secondary Duration of response according to RECIST v1.1 Approximately 3 years
Secondary Progression-free survival (PFS) according to RECIST v1.1 Approximately 3 years