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Clinical Trial Details — Status: Completed

Administrative data

NCT number NCT02547935
Other study ID # D1690C00023
Secondary ID
Status Completed
Phase Phase 2/Phase 3
First received
Last updated
Start date September 21, 2015
Est. completion date May 18, 2018

Study information

Verified date July 2019
Source AstraZeneca
Contact n/a
Is FDA regulated No
Health authority
Study type Interventional

Clinical Trial Summary

The purpose of this clinical research study is to determine whether dapagliflozin alone or in combination with saxagliptin can decrease albuminuria and improve glycemic control in patients with Type 2 diabetes, albuminuria and renal impairment (CKD). The study is planned to randomize a total of 450 patients (150 patients per treatment arm)


Recruitment information / eligibility

Status Completed
Enrollment 459
Est. completion date May 18, 2018
Est. primary completion date May 18, 2018
Accepts healthy volunteers No
Gender All
Age group 18 Years to 130 Years
Eligibility Inclusion Criteria:

- Provision of informed consent prior to any study specific procedures

- Female or male aged =18 years

- History of type 2 diabetes mellitus for more than 12 months

- HbA1c=7.0% and =11.0%

- Stable antidiabetic treatment during the last 12 weeks up to randomization

- eGFR 25-75 mL/minute/1.73m2, inclusive

- Micro or macroalbuminuria (UACR 30 - 3500 mg/g)

- Treatment with ACE inhibitor or an ARB for at least 3 months prior to screening

- Body mass index between 20 and 45 kg/m2

Exclusion Criteria:

- Any of the following CV/Vascular Diseases within 3 month prior to signing the consent at Visit 1:

- Myocardial infarction

- cardiac surgery or revascularization (CABG/PTCA)

- unstable angina

- unstable HF

- New York Heart Association (NYHA) Class III-IV

- transient ischemic attack (TIA) or significant cerebrovascular disease

- unstable or previously undiagnosed arrhythmia

- Significant hepatic disease, including, but not limited to, chronic active hepatitis and/or severe hepatic insufficiency

- Aspartate Aminotransferase (AST) or Alanine Aminotransferase (ALT) > 3X ULN

- Total Bilirubin (TB) >2 mg/dL (34.2 µmol/L)

- History of acute kidney injury requiring renal replacement therapy (dialysis or ultrafiltration) or any biopsy or imaging verifying intercurrent kidney disease other than diabetic nephropathy or diabetic nephropathy with nephrosclerosis

- Ongoing treatment with a SGLT2 inhibitor, GLP-1 agonist or DPP4 inhibitors

- Any condition which, in the judgment of the Investigator, may render the patient unable to complete the study or which may pose a significant risk to the patient or patient suspected or with confirmed poor protocol or medication compliance

Study Design


Related Conditions & MeSH terms


Intervention

Drug:
Dapagliflozin 10 mg
Tablets administered orally once daily for 24 weeks.
Saxagliptin 2.5 mg
Tablets administered orally once daily for 24 weeks.
Matching Placebo for Dapagliflozin 10 mg and Saxagliptin 2.5mg
Tablets administered orally once daily for 24 weeks.

Locations

Country Name City State
Australia Research Site Box Hill
Australia Research Site Campbelltown
Australia Research Site Geelong
Australia Research Site Herston
Canada Research Site Ajax Ontario
Canada Research Site Cambridge Ontario
Canada Research Site Chicoutimi Quebec
Canada Research Site Moncton New Brunswick
Canada Research Site Quebec
Canada Research Site Saint-Jerome Quebec
Canada Research Site Scarborough Ontario
Canada Research Site Scarborough Ontario
Canada Research Site Sherbrooke Quebec
Canada Research Site Toronto Ontario
Canada Research Site Winnipeg Manitoba
Japan Research Site Chuo-ku
Japan Research Site Chuo-ku
Japan Research Site Chuo-ku
Japan Research Site Hachioji-shi
Japan Research Site Higashiosaka-shi
Japan Research Site Kisarazu-shi
Japan Research Site Kyoto-shi
Japan Research Site Neyagawa-shi
Japan Research Site Nishinomiya-shi
Japan Research Site Oita-shi
Japan Research Site Osaka-shi
Japan Research Site Osaka-shi
Japan Research Site Sendai-shi
Japan Research Site Shinjuku-ku
Japan Research Site Toyonaka-shi
Korea, Republic of Research Site Ansan-si
Korea, Republic of Research Site Busan
Korea, Republic of Research Site Cheongju-si
Korea, Republic of Research Site Daejeon
Korea, Republic of Research Site Seongnam-si
Korea, Republic of Research Site Seoul
Korea, Republic of Research Site Seoul
Korea, Republic of Research Site Seoul
Korea, Republic of Research Site Suwon-si
Korea, Republic of Research Site Wonju-si
Mexico Research Site Aguascalientes
Mexico Research Site Guadalajara
Mexico Research Site Guadalajara
Mexico Research Site Guadalajara
Mexico Research Site Mexico
Mexico Research Site Mexico
Mexico Research Site México
Mexico Research Site Monterey
Mexico Research Site Monterrey
Mexico Research Site Monterrey
Mexico Research Site Queretaro
Mexico Research Site Zapopan
Mexico Research Site Zapopan, Jalisco
South Africa Research Site Benoni
South Africa Research Site Cape Town
South Africa Research Site Cape Town
South Africa Research Site Durban
South Africa Research Site Kuilsrivier
South Africa Research Site Mamelodi East
South Africa Research Site Muckleneuk
South Africa Research Site Paarl
South Africa Research Site Pretoria
Spain Research Site A Coruña
Spain Research Site Barcelona
Spain Research Site Madrid
Spain Research Site Sabadell (Barcelona)
Spain Research Site Santiago(A Coruña)
Spain Research Site Valencia
Taiwan Research Site Changhua
Taiwan Research Site Kaohsiung Hsien
Taiwan Research Site New Taipei
Taiwan Research Site New Taipei City
Taiwan Research Site Taichung
Taiwan Research Site Taipei City
Taiwan Research Site Yong-Kang City
United States Research Site Augusta Georgia
United States Research Site Bangor Maine
United States Research Site Bronx New York
United States Research Site Brownsville Texas
United States Research Site Burke Virginia
United States Research Site Chicago Illinois
United States Research Site Chula Vista California
United States Research Site Concord California
United States Research Site Cypress Texas
United States Research Site El Centro California
United States Research Site Greensboro North Carolina
United States Research Site Greenville South Carolina
United States Research Site Hollywood Florida
United States Research Site Houston Texas
United States Research Site Kansas City Missouri
United States Research Site La Mesa California
United States Research Site Las Vegas Nevada
United States Research Site Long Beach California
United States Research Site Los Gatos California
United States Research Site Meridian Idaho
United States Research Site Miami Florida
United States Research Site Morehead City North Carolina
United States Research Site New Port Richey Florida
United States Research Site North Hollywood California
United States Research Site Palm Harbor Florida
United States Research Site Peoria Arizona
United States Research Site Philadelphia Pennsylvania
United States Research Site Pompano Beach Florida
United States Research Site Richmond Virginia
United States Research Site Riverside California
United States Research Site Rocky Mount North Carolina
United States Research Site Salt Lake City Utah
United States Research Site San Antonio Texas
United States Research Site San Diego California
United States Research Site San Dimas California
United States Research Site Springfield Gardens New York
United States Research Site Sugar Land Texas

Sponsors (1)

Lead Sponsor Collaborator
AstraZeneca

Countries where clinical trial is conducted

United States,  Australia,  Canada,  Japan,  Korea, Republic of,  Mexico,  South Africa,  Spain,  Taiwan, 

Outcome

Type Measure Description Time frame Safety issue
Primary Adjusted Mean Change From Baseline in Glycosylated Haemoglobin (HbA1c): Comparison of Dapagliflozin 10 mg Plus Saxagliptin 2.5 mg and Placebo at Week 24 HbA1c was analysed at baseline and every 4 weeks during the 24-week treatment period. Only measurements prior to rescue or treatment discontinuation were analysed. The adjusted mean change from baseline at Week 24 was analysed using a mixed model repeated measures (MMRM) model. Baseline and Week 24
Primary Adjusted Mean Percent Change From Baseline in Urine Albumin-to-Creatinine Ratio (UACR) at Week 24 UACR was analysed at baseline and every 4 weeks during the 24-week treatment period. All measurements regardless of rescue medication or treatment discontinuation were analysed. UACR values were first transformed to logarithms and the results were based on exponentiation of model estimates and expressed as adjusted mean percent change from baseline at Week 24. Baseline and Week 24
Secondary Adjusted Mean Percent Change From Baseline in Total Body Weight at Week 24 Total body weight was measured in kilograms (kg) at baseline and at Week 1 then every 4 weeks during the 24-week treatment period. All measurements regardless of rescue medication or treatment discontinuation were analysed. Total body weight values were first transformed to logarithms and the results were based on exponentiation of model estimates and expressed as adjusted mean percent change from baseline at Week 24. Baseline and Week 24
Secondary Adjusted Mean Change From Baseline in Fasting Plasma Glucose (FPG) at Week 24 FPG was analysed at baseline and Week 1 then every 4 weeks during the 24-week treatment period. Only measurements prior to rescue or treatment discontinuation were analysed. The adjusted mean change from baseline at Week 24 was analysed using a MMRM model. Baseline and Week 24
Secondary Percentage of Patients Achieving at Least 30% Reduction in UACR at Week 24 The percentage of patients meeting the criteria of at least a 30% reduction in UACR, was analysed using a logistic regression model. If no measurement was available at Week 24 the last available post-baseline measurement was carried forward (Last Observation Carried Forward [LOCF]). From baseline up to Week 24
Secondary Percentage of Patients Achieving a Reduction in HbA1c of Less Than 7.0% at Week 24 The percentage of patients meeting the criteria of a less than 7% reduction in HbA1c, was analysed using a logistic regression model. If no measurement was available at Week 24 the last available post-baseline measurement was carried forward (LOCF). Only measurements prior to rescue or treatment discontinuation were analysed. From baseline to Week 24
Secondary Adjusted Mean Change From Baseline in Seated Systolic Blood Pressure (SBP) at Week 24 Seated SBP was analysed at baseline, Week 1 and every 4 weeks during the 24-week treatment period. All measurements regardless of rescue medication or treatment discontinuation were analysed. The adjusted mean change from baseline at Week 24 was analysed using a MMRM model. Baseline and Week 24
Secondary Adjusted Mean Change From Baseline in HbA1c: Comparison of Dapagliflozin 10 mg and Placebo at Week 24 HbA1c was analysed at baseline and every 4 weeks during the 24-week treatment period. Only measurements prior to rescue or treatment discontinuation were analysed. The adjusted mean change from baseline at Week 24 was analysed using a MMRM model. Baseline and Week 24