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Clinical Trial Details — Status: Completed

Administrative data

NCT number NCT00975182
Other study ID # GDC4626g
Secondary ID GO01301
Status Completed
Phase Phase 1
First received September 8, 2009
Last updated November 1, 2016
Start date September 2009
Est. completion date September 2014

Study information

Verified date November 2016
Source Genentech, Inc.
Contact n/a
Is FDA regulated No
Health authority United States: Food and Drug Administration
Study type Interventional

Clinical Trial Summary

This is an open-label, multicenter, Phase Ib dose-escalation study to assess the safety, tolerability, and pharmacokinetics (PK) of oral (PO) GDC-0941 administered in combination with PO erlotinib in patients with advanced solid tumors and patients with locally advanced or metastatic non-small cell lung cancer (NSCLC) who have failed at least one prior chemotherapy regimen.


Recruitment information / eligibility

Status Completed
Enrollment 58
Est. completion date September 2014
Est. primary completion date September 2014
Accepts healthy volunteers No
Gender Both
Age group 18 Years and older
Eligibility Inclusion Criteria:

- Documented locally advanced or metastatic solid tumors for which standard therapy either does not exist or has proven ineffective or intolerable (dose-escalation stage only)

- Documented locally advanced or metastatic NSCLC in patients who have failed at least one prior chemotherapy-based regimen for incurable disease (cohort-expansion stage only)

- Adequate organ function as assessed by laboratory tests

- Evaluable disease or disease measurable per Response Evaluation Criteria in Solid Tumors (RECIST)

- Agreement to use an effective form of contraception for the duration of the study

Exclusion Criteria:

- Any anti-cancer therapy (e.g., chemotherapy, biologic therapy, or hormonal therapy) within a specified timeframe prior to first study treatment

- Prior treatment with PI3K pathway-inhibiting agents (cohort-expansion stage only)

- History of Grade >= 3 fasting hyperglycemia or diabetes requiring regular medication

- Current clinically significant and uncontrolled systemic disease (e.g., cardiovascular, pulmonary, or metabolic)

- History of clinically significant cardiac or pulmonary dysfunction

- History of malabsorption syndrome or other condition that would interfere with enteral absorption

- Clinically significant history of liver disease

- Any condition requiring full-dose anticoagulants, such as warfarin, heparin, or thrombolytic agents

- Active autoimmune disease and/or need for corticosteroid therapy

- Known brain metastases that are untreated, symptomatic, or require therapy

- Pregnancy, lactation, or breastfeeding

Study Design

Allocation: Non-Randomized, Intervention Model: Single Group Assignment, Masking: Open Label, Primary Purpose: Treatment


Related Conditions & MeSH terms


Intervention

Drug:
GDC-0941
Oral repeating dose
erlotinib HCl
Oral repeating dose

Locations

Country Name City State
n/a

Sponsors (1)

Lead Sponsor Collaborator
Genentech, Inc.

Countries where clinical trial is conducted

United States,  Netherlands, 

Outcome

Type Measure Description Time frame Safety issue
Primary Incidence, nature, and severity of adverse events Through study completion or early study discontinuation No
Primary Tumor response Assessed at periodic intervals No
Secondary PK parameters of GDC-0941 (total exposure, and maximum and minimum serum concentrations) Through study completion or early study discontinuation No