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Clinical Trial Details — Status: Completed

Administrative data

NCT number NCT01186861
Other study ID # OSI-906-205
Secondary ID 2010-020916-12
Status Completed
Phase Phase 2
First received
Last updated
Start date March 4, 2011
Est. completion date March 11, 2015

Study information

Verified date August 2018
Source Astellas Pharma Inc
Contact n/a
Is FDA regulated No
Health authority
Study type Interventional

Clinical Trial Summary

A multicenter, randomized, double-blind, placebo-controlled, phase 2 study with a 1:1 randomization scheme.


Description:

Adult patients with advanced Non-small Cell Lung Cancer (NSCLC) and nonprogression after platinum-based chemotherapy will be randomized 1:1 to receive either OSI-906 plus erlotinib or placebo plus erlotinib.


Recruitment information / eligibility

Status Completed
Enrollment 205
Est. completion date March 11, 2015
Est. primary completion date July 1, 2013
Accepts healthy volunteers No
Gender All
Age group 18 Years and older
Eligibility Inclusion Criteria:

- Histologically confirmed locally advanced or metastatic stage IIIB or IV NSCLC

- Have experienced Complete Response (CR), Partial Response (PR) or Stable Disease (SD) following completion of 4 cycles of first-line platinum-based chemotherapy and are not progressing at time of entry into study (prior completed first-line combination bevacizumab therapy is permitted; however, current use of maintenance bevacizumab is not permitted. A maximum interval of 28 days between the last day of the treatment cycle and randomization

- Patient has recovered from prior chemotherapy-related toxicity to = grade 2

- EGFR mutation status must be confirmed for participation in the study. EGFR analysis can be performed either by central or local laboratory. If analysis is done locally, verifiable documentation confirming the EGFR mutation status must be submitted for review and approval by APGD prior to randomization. If no local result is available, formalin-fixed, paraffin-embedded archival tissue representative of the tumor or in the absence of archival tissue, a fresh tumor tissue sample of sufficient size to perform EGFR mutation analysis must be submitted centrally. Results of the central analysis must be available prior to randomization. Additionally, subjects should provide tissue blocks centrally for biomarker analysis whenever possible. Ideal tissue requirement: block with =5 mm2 tumor area sufficient to provide four 4-micron, and five 10-micron sections)

- Measurable disease (for those patients with PR or SD after first-line platinum-based chemotherapy) according to Response Evaluation Criteria in Solid Tumors (RECIST) (version 1.1)

- Eastern Cooperative Oncology Group (ECOG) Performance Status(PS) 0 - 1

- Previous adjuvant or neo-adjuvant treatment is permitted

- Must be able to take oral medication

- Fasting glucose = 150 mg/dL (8.3 mmol/L). Concurrent use of non-insulinotropic antihyperglycemic therapy is permitted if the dose has been stable for = 4 weeks at the time of randomization

- Adequate hematopoietic, hepatic, and renal function defined as follows:

- Neutrophil count = 1.5 x 109/L

- Platelet count = 100 x 109/L

- Bilirubin = 1.5 x Upper Limit of Normal (ULN)

- AST and ALT = 2.5 x ULN, or = 5 x ULN if patient has documented liver metastases

- Serum creatinine = 1.5 x ULN

- Potassium, magnesium and calcium within normal limits (supplementation and retesting is permitted)

Female patient must be either:

- Of non child bearing potential:

- post-menopausal (defined as at least 1 year without any menses) prior to

Screening, or

- documented surgically sterile or status post hysterectomy (at least 1 month prior to Screening)

- Or, if of childbearing potential:

- must have a negative urine pregnancy test at Screening, and

- must use two forms of birth control (one of which must be a barrier method) starting at Screening and throughout the study period and for 30 days after final study drug administration

- Female patient must not be breastfeeding at Screening or during the study period and for 30 days after final study drug administration

- Female patient must not donate ova starting at Screening and throughout the study period and for 30 days after final study drug administration

- Male patient and their female spouse/partners who are of childbearing potential must be using highly effective contraception consisting of two forms of birth control (one of which must be a barrier method) starting at Screening and continue throughout the study period and for 30 days after final study drug administration

- Male patient must not donate sperm starting at Screening and throughout the study period and for at least 30 days after final study drug administration

- Prior radiation therapy is permitted provided patients have recovered from acute toxic effects of radiotherapy prior to randomization. A minimum of 28 days must have elapsed between the end of radiotherapy and randomization

- Prior surgery is permitted provided that the surgery was performed 21 days prior to randomization and adequate wound healing has occurred prior to randomization

- Patients must provide written (signed) informed consent to participate in the study and for use of tumor tissues

Exclusion Criteria:

- Prior exposure to agents directed at the Human Epidermal Receptor (HER) axis (eg, erlotinib, gefitinib, cetuximab, and trastuzumab)

- Malignancies other than NSCLC within past 3 years (exceptions if curatively treated: basal or squamous cell carcinoma of skin; locally advanced prostate cancer; ductal carcinoma in situ of breast; in situ cervical carcinoma; and superficial bladder cancer)

- Type 1 diabetes mellitus or Type 2 diabetes mellitus currently requiring insulinotropic or insulin therapy

- Prior insulin-like growth factor receptor (IGF-1R)

- Prior investigational agent within 21 days prior to randomization

- Concurrent use of maintenance bevacizumab

- History of poorly controlled gastrointestinal disorders that could affect the absorption of study drug (eg, Crohn's disease, ulcerative colitis, etc)

- History (within last 180 days) of significant cardiovascular disease unless the disease is well-controlled. Significant cardiac disease includes second/third degree heart block; clinically significant ischemic heart disease; superior vena cava (SVC) syndrome; poorly controlled hypertension; congestive heart failure of New York Heart Association (NYHA) Class II or worse (slight limitation of physical activity; comfortable at rest, but ordinary physical activity results in fatigue, palpitation, or dyspnea)

- History of arrhythmia (multifocal premature ventricular contractions [PVCs], bigeminy, trigeminy, ventricular tachycardia, or uncontrolled atrial fibrillation) that is symptomatic or requires treatment (= grade 3), left bundle branch block (LBBB), or asymptomatic sustained ventricular tachycardia are not allowed. Patients with atrial fibrillation controlled by medication are not excluded

- Mean QTcF interval > 450 msec based on independent central reviewer analysis of screening visit ECGs

- Use of drugs that have a known risk of causing Torsades de Pointes (TdP) are prohibited within 14 days prior to randomization

- Use of the potent CYP1A2 inhibitors ciprofloxacin and fluvoxamine. Other less potent CYP1A2 inhibitors/inducers are not excluded

- Use of potent CYP3A4 inhibitor such as ketoconazole, clarithromycin, atazanavir, indinavir, itraconazole, nefazodone, nelfinavir, ritonavir, saquinavir, telithromycin, troleandomycin (TAO), or voriconazole

- Use of proton pump inhibitors such as omeprazole. Use of H2-receptor antagonists such as ranitidine are not excluded

- History of cerebrovascular accident (CVA) within 180 days prior to randomization or that resulted in ongoing neurologic instability

- Active infection, serious underlying medical condition (including any type of active seizure disorder within 12 months prior to randomization), or serious chronic illness that would impair the ability of the patient to receive study drug

- History of any psychiatric or neurologic condition that might impair the patient's ability to understand or to comply with the requirements of the study or to provide informed consent

- Pregnant or breast-feeding females

- Symptomatic brain metastases that are not stable, require steroids, or that have required radiation and/or other related treatment (e.g., anti-epileptic medication) within 21 days prior to randomization

- History of allergic reactions attributed to compounds of similar chemical or biologic composition to study drug

- Participated in any interventional clinical study or has been treated with any investigational drugs within 30 days or 5 half lives whichever is longer, prior to the initiation of Screening or during the course of the study

Study Design


Related Conditions & MeSH terms


Intervention

Drug:
OSI-906
Tablet administered with food and with up to 200 mL of water
erlotinib
Tablet administered at least 2 hours after food with up to 200 mL of water
placebo
Tablet administered at least 2 hours after food with up to 200 mL of water

Locations

Country Name City State
Brazil Site BR55005 Barretos
Brazil Site BR55004 Brasilia
Brazil Site BR55015 Cachoeiro de Itapemirim
Brazil Site BR55011 Florianopolis
Brazil Site BR55003 Fortaleza
Brazil Site BR55016 Goiania
Brazil Site BR55006 Ijui
Brazil Site BR55001 Itajai
Brazil Site BR55008 Piracicaba
Brazil Site BR55013 Porto Alegre
Brazil Site BR55014 Porto Alegre
Brazil Site BR55012 Ribeirao Preto
Brazil Site BR55002 Rio de Janeiro
Brazil Site BR55007 Sao Paulo
Canada Site CA11001 Oshawa
Canada Site CA11004 Ottawa
Canada Site CA11002 Toronto
Canada Site CA11006 Toronto
Germany Site DE49014 Berlin
Germany Site DE49011 Dortmund
Germany Site DE49003 Grosshansdorf
Germany Site DE49001 Heidelberg
Germany Site DE49002 Hemer
Germany Site DE49009 Homburg/Saar
Germany Site DE49006 Immenhausen
Germany Site DE49012 Karlsruhe
Germany Site DE49015 Kassel
Germany Site DE49008 Koln
Germany Site DE49010 Lubeck
Germany Site DE49013 Mainz
Germany Site DE49005 Minden
Korea, Republic of Site KR82007 Busan
Korea, Republic of Site KR82006 Hwasun
Korea, Republic of Site KR82008 Incheon
Korea, Republic of Site KR82004 Seongnam-si
Korea, Republic of Site KR82002 Seoul
Korea, Republic of Site KR82003 Seoul
Korea, Republic of Site KR82005 Seoul
Korea, Republic of Site KR82001 Suwon
Poland Site PL48002 Elblag
Poland Site PL48005 Szczecin
Poland Site PL48008 Torun
Poland Site PL48006 Wroclaw
Romania Site RO40005 Alba Iulia
Romania Site RO40001 Baia Mare
Romania Site RO40007 Brasov
Romania Site RO40002 Cluj-Napoca
Romania Site RO40003 Cluj-Napoca
Romania Site RO40006 Craiova
Romania Site RO40004 Hunedoara
Russian Federation Site RU70002 Chelaybinsk
Russian Federation Site RU70010 Kazan
Russian Federation Site RU70007 Saint Petersburg
Russian Federation Site RU70009 Saint Petersburg
Russian Federation Site RU70011 Saint Petersburg
United Kingdom Site GB44007 Bristol
United Kingdom Site GB44006 Dundee
United Kingdom Site GB44003 Leeds
United Kingdom Site GB44002 Leicester
United Kingdom Site GB44005 London
United Kingdom Site GB44001 Manchester
United Kingdom Site GB44004 Southampton
United States Site US10002 Albany Georgia
United States Site US10008 Chicago Illinois
United States Site US10004 Greensboro North Carolina
United States Site US10007 Jacksonville Florida
United States Site US10001 Port Saint Lucie Florida
United States Site US10011 Scarborough Maine
United States Site US10010 Winston-Salem North Carolina

Sponsors (1)

Lead Sponsor Collaborator
Astellas Pharma Inc

Countries where clinical trial is conducted

United States,  Brazil,  Canada,  Germany,  Korea, Republic of,  Poland,  Romania,  Russian Federation,  United Kingdom, 

Outcome

Type Measure Description Time frame Safety issue
Primary The Progression Free Survival (PFS) of maintenance OSI-906 plus erlotinib, or placebo plus erlotinib in patients with nonprogression following four cycles of first-line platinum-based chemotherapy for advanced NSCLC in the overall population PFS is defined as the time from randomization to disease progression based on RECIST v1.1 or death due to any cause whichever comes first 22 months
Secondary Overall survival (OS) The time from the date of randomization until the documented date of death 27 months
Secondary Disease control Rate (DCR) The proportion of patients with a best overall response of continued Complete Response (CR), CR, Partial Response (PR), OR Stable Disease (SD) based on RECIST criteria 27 months
Secondary Best overall response rate (ORR) The proportion of patients with a best overall response of CR or PR based on RECIST criteria 27 months
Secondary Response upgrade rate (RUR) The proportion of patients with a response upgrade 27 months
Secondary Duration of response The time from the date of the first documented response (CR/PR) to documented progression or death due to underlying cancer 27 months
Secondary Safety assessed through physical examination, vital signs, clinical laboratory tests, electrocardiograms (ECG) and Adverse Events 27 months